Assay Detail
Functional
CHEMBL4403391
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Antiparasitic activity against Plasmodium falciparum W2
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Plasmodium falciparum |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
New dimensions in the field of antimalarial research against malaria resurgence.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 8.08 | 8.87 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3264503 | — | — | 1 | 8.87 |
| CHEMBL3264171 | — | — | 1 | 8.58 |
| CHEMBL3264174 | — | — | 1 | 8.58 |
| CHEMBL3264178 | — | — | 1 | 8.58 |
| CHEMBL3264179 | — | — | 1 | 8.58 |
| CHEMBL3264183 | — | — | 1 | 8.58 |
| CHEMBL3264190 | — | — | 1 | 8.58 |
| CHEMBL3264192 | — | — | 1 | 8.58 |
| CHEMBL3264501 | — | — | 1 | 8.43 |
| CHEMBL4555605 | — | — | 1 | 6.95 |
| CHEMBL4446072 | — | — | 1 | 6.43 |
| CHEMBL76 | CHLOROQUINE | 4.0 | 1 | 6.16 |
| CHEMBL197308 | FERRUGINOL | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3264503 | — | IC50 | = | 1.35 | nM | 8.87 |
| CHEMBL3264171 | — | IC50 | = | 2.63 | nM | 8.58 |
| CHEMBL3264174 | — | IC50 | = | 2.63 | nM | 8.58 |
| CHEMBL3264178 | — | IC50 | = | 2.63 | nM | 8.58 |
| CHEMBL3264179 | — | IC50 | = | 2.63 | nM | 8.58 |
| CHEMBL3264183 | — | IC50 | = | 2.63 | nM | 8.58 |
| CHEMBL3264190 | — | IC50 | = | 2.63 | nM | 8.58 |
| CHEMBL3264192 | — | IC50 | = | 2.63 | nM | 8.58 |
| CHEMBL3264501 | — | IC50 | = | 3.74 | nM | 8.43 |
| CHEMBL4555605 | — | IC50 | = | 112.5 | nM | 6.95 |
| CHEMBL4446072 | — | IC50 | = | 370.0 | nM | 6.43 |
| CHEMBL76 | CHLOROQUINE | IC50 | = | 697.94 | nM | 6.16 |
| CHEMBL197308 | FERRUGINOL | IC50 | = | 0.9 | ug.mL-1 | - |