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Assay Detail

CHEMBL4403436

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human PC3 cells assessed as reduction in cell viability
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type PC-3
Confidence 1 — Organism
Curated By Autocuration

Target

PC-3 (CHEMBL390)
Type CELL-LINE
Organism Homo sapiens

Publication

Recent advances in α,β-unsaturated carbonyl compounds as mitochondrial toxins.
Hossain M, Das U, Dimmock JR.
Eur J Med Chem (2019) 183 : 111687 -111687
PubMed 31539776 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.09 5.09

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL317469 1 5.09
CHEMBL105310 2',4'-DIHYDROXYCHALCONE 1 5.09
CHEMBL4514458 1 5.09
CHEMBL4537198 1 5.09
CHEMBL4447825 1 5.09

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL317469 IC50 = 8080.0 nM 5.09
CHEMBL105310 2',4'-DIHYDROXYCHALCONE IC50 = 8080.0 nM 5.09
CHEMBL4514458 IC50 = 8080.0 nM 5.09
CHEMBL4537198 IC50 = 8080.0 nM 5.09
CHEMBL4447825 IC50 = 8080.0 nM 5.09