Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4403520

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiparasitic activity against Toxoplasma gondii infected in human HFF cells after 4 hrs
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Toxoplasma gondii
Confidence 1 — Organism
Curated By Autocuration

Target

Toxoplasma gondii (CHEMBL612888)
Type ORGANISM
Organism Toxoplasma gondii

Publication

Recent progress on anti-Toxoplasma drugs discovery: Design, synthesis and screening.
Deng Y, Wu T, Zhai SQ, Li CH.
Eur J Med Chem (2019) 183 : 111711 -111711
PubMed 31585276 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 6.34 6.89

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4525036 1 6.89
CHEMBL4571126 1 6.70
CHEMBL591128 1 6.57
CHEMBL601497 1 5.89
CHEMBL527577 1 5.64

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4525036 IC50 = 130.0 nM 6.89
CHEMBL4571126 IC50 = 200.0 nM 6.70
CHEMBL591128 IC50 = 270.0 nM 6.57
CHEMBL601497 IC50 = 1300.0 nM 5.89
CHEMBL527577 IC50 = 2300.0 nM 5.64