Assay Detail
Binding
CHEMBL4404876
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Agonist activity at rat FFA3 receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Structure-Activity Relationship Studies of Tetrahydroquinolone Free Fatty Acid Receptor 3 Modulators.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 6.20 | 6.39 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4530642 | — | — | 1 | 6.39 |
| CHEMBL4564389 | — | — | 1 | 6.34 |
| CHEMBL4448591 | — | — | 1 | 5.87 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4530642 | — | EC50 | = | 407.38 | nM | 6.39 |
| CHEMBL4564389 | — | EC50 | = | 457.09 | nM | 6.34 |
| CHEMBL4448591 | — | EC50 | = | 1348.96 | nM | 5.87 |