Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4408790

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Competitive irreversible inhibition of CDK14/cyclin Y (unknown origin) in presence of Km ATP
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 7 — Homologous single protein target
Curated By Autocuration

Target

Cyclin-dependent kinase 14/Cyclin-Y (CHEMBL4296115)
Type PROTEIN COMPLEX
Organism Homo sapiens

Publication

Cyclin dependent kinase (CDK) inhibitors as anticancer drugs: Recent advances (2015-2019).
Sánchez-Martínez C, Lallena MJ, Sanfeliciano SG, de Dios A.
Bioorg Med Chem Lett (2019) 29 : 126637 -126637
PubMed 31477350 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.06 7.06

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4580787 1 7.06

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4580787 IC50 = 88.0 nM 7.06