Assay Detail
Binding
CHEMBL4409301
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Binding affinity to kappa opioid receptor (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Progress in the development of more effective and safer analgesics for pain management.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 8.96 | 9.23 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2381583 | 22-THIOCYANATOSALVINORIN A | — | 1 | 9.23 |
| CHEMBL4464797 | — | — | 1 | 8.68 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2381583 | 22-THIOCYANATOSALVINORIN A | Kd | = | 0.59 | nM | 9.23 |
| CHEMBL4464797 | — | Kd | = | 2.1 | nM | 8.68 |