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Assay Detail

CHEMBL4409322

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Functional
Inhibition of delta opioid receptor (unknown origin) expressed in human UO5S cells by [35S]-GTPgammaS binding assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Delta-type opioid receptor (CHEMBL236)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Progress in the development of more effective and safer analgesics for pain management.
Turnaturi R, Chiechio S, Salerno L, Rescifina A, Pittalà V, Cantarella G, Tomarchio E, Parenti C, Pasquinucci L.
Eur J Med Chem (2019) 183 : 111701 -111701
PubMed 31550662 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 7.27 7.27

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1612697 1 7.27

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1612697 EC50 = 54.0 nM 7.27