Assay Detail
Binding
CHEMBL4409334
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of delta opioid receptor in guinea pig brain membranes
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Tissue | Brain |
| Subcellular | Membranes |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Progress in the development of more effective and safer analgesics for pain management.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.02 | 7.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL61630 | — | — | 1 | 7.22 |
| CHEMBL299031 | — | — | 1 | 6.81 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL61630 | — | Ki | = | 60.0 | nM | 7.22 |
| CHEMBL299031 | — | Ki | = | 155.0 | nM | 6.81 |