Assay Detail
Binding
CHEMBL4411035
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Activation of NF-KappaB (unknown origin) expressed in SH-SY5Y cells co-transfected with pNFkappaB-Luc plasmid measured after 24 hrs by Bright-Glo luciferase assay
16
Total Activities
8
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | SH-SY5Y |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Approaches for Prevention and Treatment of Neurodegenerative Diseases: ALS and Alzheimer's.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 8 | 6.22 | 6.80 |
| ECmax | 8 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4535691 | — | — | 2 | 6.80 |
| CHEMBL528694 | — | — | 2 | 6.68 |
| CHEMBL4465283 | — | — | 2 | 6.40 |
| CHEMBL1370490 | — | — | 2 | 6.30 |
| CHEMBL4474207 | — | — | 2 | 6.15 |
| CHEMBL4588896 | — | — | 2 | 5.99 |
| CHEMBL4572792 | — | — | 2 | 5.92 |
| CHEMBL4476647 | — | — | 2 | 5.49 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4535691 | — | EC50 | = | 160.0 | nM | 6.80 |
| CHEMBL528694 | — | EC50 | = | 210.0 | nM | 6.68 |
| CHEMBL4465283 | — | EC50 | = | 400.0 | nM | 6.40 |
| CHEMBL1370490 | — | EC50 | = | 500.0 | nM | 6.30 |
| CHEMBL4474207 | — | EC50 | = | 710.0 | nM | 6.15 |
| CHEMBL4588896 | — | EC50 | = | 1030.0 | nM | 5.99 |
| CHEMBL4572792 | — | EC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL4476647 | — | EC50 | = | 3270.0 | nM | 5.49 |
| CHEMBL4535691 | — | ECmax | = | 42.58 | uM | - |
| CHEMBL4474207 | — | ECmax | = | 20.15 | uM | - |
| CHEMBL4572792 | — | ECmax | = | 63.18 | uM | - |
| CHEMBL4465283 | — | ECmax | = | 34.11 | uM | - |
| CHEMBL1370490 | — | ECmax | = | 26.0 | uM | - |
| CHEMBL528694 | — | ECmax | = | 40.0 | uM | - |
| CHEMBL4588896 | — | ECmax | = | 23.53 | uM | - |
| CHEMBL4476647 | — | ECmax | = | 46.45 | uM | - |