Assay Detail
Functional
CHEMBL4416180
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Antiplasmodial activity against asexual form of Plasmodium falciparum NF54 assessed as reduction in female gametocytes activation preincubated for 48 hrs followed by gametocytes activation and measured after 24 hrs by fluorescence based automated inverted microscopic analysis
38
Total Activities
38
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Plasmodium falciparum |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Development of Chemical Entities Endowed with Potent Fast-Killing Properties against <i>Plasmodium falciparum</i> Malaria Parasites.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 38 | 6.18 | 6.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4459320 | — | — | 1 | 6.72 |
| CHEMBL4531058 | — | — | 1 | 6.52 |
| CHEMBL4566588 | — | — | 1 | 6.42 |
| CHEMBL4591417 | — | — | 1 | 6.40 |
| CHEMBL4451783 | — | — | 1 | 6.39 |
| CHEMBL4473609 | — | — | 1 | 6.33 |
| CHEMBL4288103 | — | — | 1 | 6.32 |
| CHEMBL4455587 | — | — | 1 | 6.11 |
| CHEMBL4531226 | — | — | 1 | 5.97 |
| CHEMBL4459919 | — | — | 1 | 5.88 |
| CHEMBL4436765 | — | — | 1 | 4.97 |
| CHEMBL4572858 | — | — | 1 | - |
| CHEMBL4469667 | — | — | 1 | - |
| CHEMBL4583048 | — | — | 1 | - |
| CHEMBL4446024 | — | — | 1 | - |
| CHEMBL4446015 | — | — | 1 | - |
| CHEMBL4546641 | — | — | 1 | - |
| CHEMBL4572065 | — | — | 1 | - |
| CHEMBL361497 | ARTESUNATE | 4.0 | 1 | - |
| CHEMBL4516715 | — | — | 1 | - |
| CHEMBL4586918 | — | — | 1 | - |
| CHEMBL4548154 | — | — | 1 | - |
| CHEMBL4461276 | — | — | 1 | - |
| CHEMBL4449947 | — | — | 1 | - |
| CHEMBL4585479 | — | — | 1 | - |
| CHEMBL4519443 | — | — | 1 | - |
| CHEMBL4526454 | — | — | 1 | - |
| CHEMBL4513311 | — | — | 1 | - |
| CHEMBL36 | PYRIMETHAMINE | 4.0 | 1 | - |
| CHEMBL4438004 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4459320 | — | EC50 | = | 190.0 | nM | 6.72 |
| CHEMBL4531058 | — | EC50 | = | 300.0 | nM | 6.52 |
| CHEMBL4566588 | — | EC50 | = | 380.0 | nM | 6.42 |
| CHEMBL4591417 | — | EC50 | = | 400.0 | nM | 6.40 |
| CHEMBL4451783 | — | EC50 | = | 410.0 | nM | 6.39 |
| CHEMBL4473609 | — | EC50 | = | 470.0 | nM | 6.33 |
| CHEMBL4288103 | — | EC50 | = | 480.0 | nM | 6.32 |
| CHEMBL4455587 | — | EC50 | = | 780.0 | nM | 6.11 |
| CHEMBL4531226 | — | EC50 | = | 1070.0 | nM | 5.97 |
| CHEMBL4459919 | — | EC50 | = | 1310.0 | nM | 5.88 |
| CHEMBL4436765 | — | EC50 | = | 10600.0 | nM | 4.97 |
| CHEMBL4446015 | — | EC50 | - | — | - | |
| CHEMBL4464676 | — | EC50 | - | — | - | |
| CHEMBL4446024 | — | EC50 | - | — | - | |
| CHEMBL4583048 | — | EC50 | - | — | - | |
| CHEMBL4469667 | — | EC50 | - | — | - | |
| CHEMBL4572858 | — | EC50 | - | — | - | |
| CHEMBL4593717 | — | EC50 | - | — | - | |
| CHEMBL4444451 | — | EC50 | - | — | - | |
| CHEMBL4532321 | — | EC50 | - | — | - | |
| CHEMBL4460574 | — | EC50 | - | — | - | |
| CHEMBL4567664 | — | EC50 | - | — | - | |
| CHEMBL4462111 | — | EC50 | - | — | - | |
| CHEMBL4585607 | — | EC50 | - | — | - | |
| CHEMBL4546641 | — | EC50 | - | — | - | |
| CHEMBL4572065 | — | EC50 | - | — | - | |
| CHEMBL361497 | ARTESUNATE | EC50 | > | 10000.0 | nM | - |
| CHEMBL4516715 | — | EC50 | - | — | - | |
| CHEMBL4586918 | — | EC50 | - | — | - | |
| CHEMBL4548154 | — | EC50 | - | — | - | |
| CHEMBL4461276 | — | EC50 | - | — | - | |
| CHEMBL4449947 | — | EC50 | - | — | - | |
| CHEMBL4585479 | — | EC50 | - | — | - | |
| CHEMBL4519443 | — | EC50 | - | — | - | |
| CHEMBL4526454 | — | EC50 | - | — | - | |
| CHEMBL4513311 | — | EC50 | - | — | - | |
| CHEMBL36 | PYRIMETHAMINE | EC50 | > | 10000.0 | nM | - |
| CHEMBL4438004 | — | EC50 | - | — | - |