Assay Detail
Binding
CHEMBL4417894
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of RAD52 (unknown origin) assessed as effect on ssDNA annealing using ssDNA oligonucleotide by fluorescence-quenching assay
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Inhibitors of RAD52 Recombination Protein and Methods Using Same
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 17 | 5.42 | 5.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4522859 | — | — | 1 | 5.77 |
| CHEMBL1544647 | — | — | 1 | 5.70 |
| CHEMBL3186644 | — | — | 1 | 5.70 |
| CHEMBL1325721 | — | — | 1 | 5.70 |
| CHEMBL1389885 | — | — | 1 | 5.55 |
| CHEMBL3189128 | — | — | 1 | 5.54 |
| CHEMBL1389728 | — | — | 1 | 5.46 |
| CHEMBL1373317 | — | — | 1 | 5.44 |
| CHEMBL3185804 | — | — | 1 | 5.39 |
| CHEMBL1198365 | — | — | 1 | 5.37 |
| CHEMBL4463510 | — | — | 1 | 5.32 |
| CHEMBL1573779 | — | — | 1 | 5.28 |
| CHEMBL3303124 | — | — | 1 | 5.25 |
| CHEMBL606456 | — | — | 1 | 5.22 |
| CHEMBL1428009 | — | — | 1 | 5.22 |
| CHEMBL596633 | — | — | 1 | 5.17 |
| CHEMBL1514131 | — | — | 1 | 5.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4522859 | — | IC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL1544647 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL3186644 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL1325721 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL1389885 | — | IC50 | = | 2800.0 | nM | 5.55 |
| CHEMBL3189128 | — | IC50 | = | 2900.0 | nM | 5.54 |
| CHEMBL1389728 | — | IC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL1373317 | — | IC50 | = | 3600.0 | nM | 5.44 |
| CHEMBL3185804 | — | IC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL1198365 | — | IC50 | = | 4300.0 | nM | 5.37 |
| CHEMBL4463510 | — | IC50 | = | 4800.0 | nM | 5.32 |
| CHEMBL1573779 | — | IC50 | = | 5200.0 | nM | 5.28 |
| CHEMBL3303124 | — | IC50 | = | 5600.0 | nM | 5.25 |
| CHEMBL606456 | — | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL1428009 | — | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL596633 | — | IC50 | = | 6800.0 | nM | 5.17 |
| CHEMBL1514131 | — | IC50 | = | 9800.0 | nM | 5.01 |