Assay Detail
Functional
CHEMBL4418233
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity in human OPM2 cells incubated for 48 hrs by MTT assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | OPM-2 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Inhibitors of mtor-deptor interactions and methods of use thereof
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.96 | 6.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4077014 | — | — | 1 | 6.52 |
| CHEMBL1898589 | — | — | 1 | 5.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4077014 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL1898589 | — | IC50 | = | 4000.0 | nM | 5.40 |