Assay Detail
Binding
CHEMBL4418633
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Inhibition of KLF5 promoter activity in human DLD1 cells by luciferase reporter gene assay
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Klf5 modulators
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 34 | 5.81 | 7.27 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4462423 | — | — | 1 | 7.27 |
| CHEMBL4544912 | — | — | 1 | 7.14 |
| CHEMBL1330145 | — | — | 1 | 6.57 |
| CHEMBL4550959 | — | — | 1 | 5.51 |
| CHEMBL4557517 | — | — | 1 | 5.28 |
| CHEMBL4580899 | — | — | 1 | 4.69 |
| CHEMBL4440755 | — | — | 1 | 4.23 |
| CHEMBL4438548 | — | — | 1 | - |
| CHEMBL4560458 | — | — | 1 | - |
| CHEMBL4536846 | — | — | 1 | - |
| CHEMBL4473625 | — | — | 1 | - |
| CHEMBL4528238 | — | — | 1 | - |
| CHEMBL4475045 | — | — | 1 | - |
| CHEMBL4471214 | — | — | 1 | - |
| CHEMBL4572993 | — | — | 1 | - |
| CHEMBL4451789 | — | — | 1 | - |
| CHEMBL4528989 | — | — | 1 | - |
| CHEMBL4547056 | — | — | 1 | - |
| CHEMBL4529329 | — | — | 1 | - |
| CHEMBL4441813 | — | — | 1 | - |
| CHEMBL4445136 | — | — | 1 | - |
| CHEMBL4476690 | — | — | 1 | - |
| CHEMBL4440930 | — | — | 1 | - |
| CHEMBL4451365 | — | — | 1 | - |
| CHEMBL4555755 | — | — | 1 | - |
| CHEMBL4561430 | — | — | 1 | - |
| CHEMBL4465760 | — | — | 1 | - |
| CHEMBL4548956 | — | — | 1 | - |
| CHEMBL4552481 | — | — | 1 | - |
| CHEMBL4459729 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4462423 | — | IC50 | = | 54.0 | nM | 7.27 |
| CHEMBL4544912 | — | IC50 | = | 72.0 | nM | 7.14 |
| CHEMBL1330145 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL4550959 | — | IC50 | = | 3100.0 | nM | 5.51 |
| CHEMBL4557517 | — | IC50 | = | 5300.0 | nM | 5.28 |
| CHEMBL4580899 | — | IC50 | = | 20490.0 | nM | 4.69 |
| CHEMBL4440755 | — | IC50 | = | 59000.0 | nM | 4.23 |
| CHEMBL4473625 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4593121 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4528238 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4475045 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4471214 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4572993 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4451789 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4528989 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4547056 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4560458 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4443631 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4519313 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4523051 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4536846 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4438548 | — | IC50 | >= | 7800.0 | nM | - |
| CHEMBL4529329 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4441813 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4445136 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4476690 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4440930 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4451365 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4555755 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4561430 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4465760 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4548956 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4552481 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4459729 | — | IC50 | > | 100000.0 | nM | - |