Assay Detail
Functional
CHEMBL4419277
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Growth inhibition of human NCI-H2122 cells incubated for 3 days
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NCI-H2122 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Methods and compositions for inhibiting cnksr1
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 6 | 4.54 | 4.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4542845 | — | — | 1 | 4.58 |
| CHEMBL1422005 | — | — | 1 | 4.57 |
| CHEMBL2030270 | — | — | 1 | 4.47 |
| CHEMBL4446354 | — | — | 1 | - |
| CHEMBL4528582 | — | — | 1 | - |
| CHEMBL4576938 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4542845 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL1422005 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL2030270 | — | IC50 | = | 34000.0 | nM | 4.47 |
| CHEMBL4446354 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4528582 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4576938 | — | IC50 | > | 100000.0 | nM | - |