Assay Detail
Binding
CHEMBL4424987
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in HEK293-EBNA cell membranes after 90 mins by scintillation counting method
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Plant-Based Modulators of Endocannabinoid Signaling.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 5.46 | 5.71 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL426912 | — | — | 1 | 5.71 |
| CHEMBL463546 | — | — | 1 | 5.21 |
| CHEMBL2287715 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL426912 | — | Ki | = | 1940.0 | nM | 5.71 |
| CHEMBL463546 | — | Ki | = | 6210.0 | nM | 5.21 |
| CHEMBL2287715 | — | Ki | > | 40000.0 | nM | - |