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Assay Detail

CHEMBL4426523

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of 6-Amino-9-(2-carboxy-4-((6-(4-(4-(4-(4-(3-carboxy-6-(4-(trifluoromethyl)phenyl)-naphthalen-1-yl)phenyl)piperidin-1-yl)-butyl)-1H-1,2,3-triazol-1-yl)hexyl)carbamoyl)-phenyl)-3-iminio-5-sulfo-3H-xanthene-4-sulfonate from human P2Y14R expressed in CHO cells measured after 15 mins by flow cytometric analysis
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type CHO
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

P2Y purinoceptor 14 (CHEMBL4518)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Structure-Based Design of 3-(4-Aryl-1H-1,2,3-triazol-1-yl)-Biphenyl Derivatives as P2Y14 Receptor Antagonists.
Junker A, Balasubramanian R, Ciancetta A, Uliassi E, Kiselev E, Martiriggiano C, Trujillo K, Mtchedlidze G, Birdwell L, Brown KA, Harden TK, Jacobson KA.
J Med Chem (2016) 59 : 6149 -6168
PubMed 27331270 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 12 6.94 8.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1800685 PPTN 1 8.22
CHEMBL4454538 1 7.50
CHEMBL4441075 1 7.14
CHEMBL4472517 1 7.04
CHEMBL4465763 1 6.94
CHEMBL4458050 1 6.88
CHEMBL4587611 1 6.79
CHEMBL4462380 1 6.65
CHEMBL4568641 1 6.64
CHEMBL4443391 1 6.62
CHEMBL4554777 1 6.54
CHEMBL4558911 1 6.32

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1800685 PPTN IC50 = 6.0 nM 8.22
CHEMBL4454538 IC50 = 31.7 nM 7.50
CHEMBL4441075 IC50 = 72.4 nM 7.14
CHEMBL4472517 IC50 = 91.0 nM 7.04
CHEMBL4465763 IC50 = 115.0 nM 6.94
CHEMBL4458050 IC50 = 131.0 nM 6.88
CHEMBL4587611 IC50 = 162.0 nM 6.79
CHEMBL4462380 IC50 = 224.0 nM 6.65
CHEMBL4568641 IC50 = 228.0 nM 6.64
CHEMBL4443391 IC50 = 237.0 nM 6.62
CHEMBL4554777 IC50 = 290.0 nM 6.54
CHEMBL4558911 IC50 = 481.0 nM 6.32