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Assay Detail

CHEMBL4428369

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antileishmanial activity against Leishmania amazonensis MHOM/BR/1973/M2269 promastigotes assessed as reduction in cell viability incubated up to 72 hrs by trypan blue dye based Neubauer chamber method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Leishmania amazonensis
Confidence 1 — Organism
Curated By Autocuration

Target

Leishmania amazonensis (CHEMBL612877)
Type ORGANISM
Organism Leishmania amazonensis

Publication

Verbascoside Inhibits Promastigote Growth and Arginase Activity of Leishmania amazonensis.
Maquiaveli CC, Lucon-Júnior JF, Brogi S, Campiani G, Gemma S, Vieira PC, Silva ER.
J Nat Prod (2016) 79 : 1459 -1463
PubMed 27096224 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 4.72 4.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL444478 ACETOSIDE 2.0 1 4.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL444478 ACETOSIDE EC50 = 19000.0 nM 4.72