Assay Detail
Binding
CHEMBL4429089
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Inhibition of HCV genotype 1a replicons NS5A infected in human Huh7 cells by luciferase reporter gene assay
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Hepatitis C virus subtype 1a |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Discovery of ravidasvir (PPI-668) as a potent pan-genotypic HCV NS5A inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 26 | 9.52 | 10.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4469447 | — | — | 1 | 10.30 |
| CHEMBL4580319 | — | — | 1 | 10.30 |
| CHEMBL4473534 | — | — | 1 | 10.15 |
| CHEMBL4587166 | — | — | 1 | 10.10 |
| CHEMBL4590699 | — | — | 1 | 10.10 |
| CHEMBL4462540 | — | — | 1 | 10.00 |
| CHEMBL4446538 | — | — | 1 | 9.96 |
| CHEMBL4461107 | — | — | 1 | 9.96 |
| CHEMBL4443067 | — | — | 1 | 9.92 |
| CHEMBL4578947 | — | — | 1 | 9.89 |
| CHEMBL4562653 | — | — | 1 | 9.89 |
| CHEMBL4442791 | — | — | 1 | 9.85 |
| CHEMBL4465723 | — | — | 1 | 9.66 |
| CHEMBL4448643 | — | — | 1 | 9.64 |
| CHEMBL4537091 | — | — | 1 | 9.59 |
| CHEMBL4436038 | — | — | 1 | 9.40 |
| CHEMBL4451714 | — | — | 1 | 9.37 |
| CHEMBL4582393 | — | — | 1 | 9.22 |
| CHEMBL4435313 | — | — | 1 | 9.18 |
| CHEMBL4563619 | — | — | 1 | 9.17 |
| CHEMBL4475469 | — | — | 1 | 8.92 |
| CHEMBL4442594 | — | — | 1 | 8.89 |
| CHEMBL4467806 | — | — | 1 | 8.69 |
| CHEMBL4546536 | — | — | 1 | 8.54 |
| CHEMBL4448546 | — | — | 1 | 7.40 |
| CHEMBL4442126 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4469447 | — | EC50 | = | 0.05 | nM | 10.30 |
| CHEMBL4580319 | — | EC50 | = | 0.05 | nM | 10.30 |
| CHEMBL4473534 | — | EC50 | = | 0.07 | nM | 10.15 |
| CHEMBL4587166 | — | EC50 | = | 0.08 | nM | 10.10 |
| CHEMBL4590699 | — | EC50 | = | 0.08 | nM | 10.10 |
| CHEMBL4462540 | — | EC50 | = | 0.1 | nM | 10.00 |
| CHEMBL4446538 | — | EC50 | = | 0.11 | nM | 9.96 |
| CHEMBL4461107 | — | EC50 | = | 0.11 | nM | 9.96 |
| CHEMBL4443067 | — | EC50 | = | 0.12 | nM | 9.92 |
| CHEMBL4578947 | — | EC50 | = | 0.13 | nM | 9.89 |
| CHEMBL4562653 | — | EC50 | = | 0.13 | nM | 9.89 |
| CHEMBL4442791 | — | EC50 | = | 0.14 | nM | 9.85 |
| CHEMBL4465723 | — | EC50 | = | 0.22 | nM | 9.66 |
| CHEMBL4448643 | — | EC50 | = | 0.23 | nM | 9.64 |
| CHEMBL4537091 | — | EC50 | = | 0.26 | nM | 9.59 |
| CHEMBL4436038 | — | EC50 | = | 0.4 | nM | 9.40 |
| CHEMBL4451714 | — | EC50 | = | 0.43 | nM | 9.37 |
| CHEMBL4582393 | — | EC50 | = | 0.6 | nM | 9.22 |
| CHEMBL4435313 | — | EC50 | = | 0.66 | nM | 9.18 |
| CHEMBL4563619 | — | EC50 | = | 0.68 | nM | 9.17 |
| CHEMBL4475469 | — | EC50 | = | 1.2 | nM | 8.92 |
| CHEMBL4442594 | — | EC50 | = | 1.3 | nM | 8.89 |
| CHEMBL4467806 | — | EC50 | = | 2.03 | nM | 8.69 |
| CHEMBL4546536 | — | EC50 | = | 2.85 | nM | 8.54 |
| CHEMBL4448546 | — | EC50 | = | 39.7 | nM | 7.40 |
| CHEMBL4442126 | — | EC50 | > | 100.0 | nM | - |