Assay Detail
Binding
CHEMBL4429339
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of GST-tagged Trypanosoma brucei ERK8 expressed in Escherichia coli using recombinant myelin basic protein as substrate after 30 mins in presence of 32P-gamma-ATP by Michaelis-Menten analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Trypanosoma brucei |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery and antiparasitic activity of AZ960 as a Trypanosoma brucei ERK8 inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 5.90 | 5.90 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1774055 | — | — | 1 | 5.90 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1774055 | — | Ki | = | 1250.0 | nM | 5.90 |