Assay Detail
Binding
CHEMBL4477289
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of [3H]PDBu binding to recombinant full length human PKCdelta expressed in baculovirus expression system incubated for 5 mins by scintillation counting method
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Inhibition of Chikungunya Virus-Induced Cell Death by Salicylate-Derived Bryostatin Analogues Provides Additional Evidence for a PKC-Independent Pathway.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 22 | 7.99 | 8.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 8.96 |
| CHEMBL4565484 | — | — | 1 | 8.89 |
| CHEMBL4533216 | — | — | 1 | 8.72 |
| CHEMBL4574406 | — | — | 1 | 8.57 |
| CHEMBL4593581 | — | — | 1 | 8.55 |
| CHEMBL4536091 | — | — | 1 | 8.48 |
| CHEMBL4526756 | — | — | 1 | 8.47 |
| CHEMBL4576842 | — | — | 1 | 8.44 |
| CHEMBL4525186 | — | — | 1 | 8.40 |
| CHEMBL4574986 | — | — | 1 | 8.36 |
| CHEMBL4550131 | — | — | 1 | 8.29 |
| CHEMBL4542079 | — | — | 1 | 8.23 |
| CHEMBL4560593 | — | — | 1 | 8.12 |
| CHEMBL4535813 | — | — | 1 | 8.10 |
| CHEMBL4564420 | — | — | 1 | 8.04 |
| CHEMBL4519769 | — | — | 1 | 7.92 |
| CHEMBL4541641 | — | — | 1 | 7.75 |
| CHEMBL4559327 | — | — | 1 | 7.55 |
| CHEMBL4575057 | — | — | 1 | 6.06 |
| CHEMBL4212128 | — | — | 1 | 6.00 |
| CHEMBL4482943 | — | — | 1 | 5.92 |
| CHEMBL4550478 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL449158 | BRYOSTATIN 1 | Ki | = | 1.1 | nM | 8.96 |
| CHEMBL4565484 | — | Ki | = | 1.3 | nM | 8.89 |
| CHEMBL4533216 | — | Ki | = | 1.9 | nM | 8.72 |
| CHEMBL4574406 | — | Ki | = | 2.7 | nM | 8.57 |
| CHEMBL4593581 | — | Ki | = | 2.8 | nM | 8.55 |
| CHEMBL4536091 | — | Ki | = | 3.3 | nM | 8.48 |
| CHEMBL4526756 | — | Ki | = | 3.4 | nM | 8.47 |
| CHEMBL4576842 | — | Ki | = | 3.6 | nM | 8.44 |
| CHEMBL4525186 | — | Ki | = | 4.0 | nM | 8.40 |
| CHEMBL4574986 | — | Ki | = | 4.4 | nM | 8.36 |
| CHEMBL4550131 | — | Ki | = | 5.1 | nM | 8.29 |
| CHEMBL4542079 | — | Ki | = | 5.9 | nM | 8.23 |
| CHEMBL4560593 | — | Ki | = | 7.6 | nM | 8.12 |
| CHEMBL4535813 | — | Ki | = | 7.9 | nM | 8.10 |
| CHEMBL4564420 | — | Ki | = | 9.1 | nM | 8.04 |
| CHEMBL4519769 | — | Ki | = | 12.0 | nM | 7.92 |
| CHEMBL4541641 | — | Ki | = | 18.0 | nM | 7.75 |
| CHEMBL4559327 | — | Ki | = | 28.0 | nM | 7.55 |
| CHEMBL4575057 | — | Ki | = | 880.0 | nM | 6.06 |
| CHEMBL4212128 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL4482943 | — | Ki | = | 1200.0 | nM | 5.92 |
| CHEMBL4550478 | — | Ki | > | 250.0 | nM | - |