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Assay Detail

CHEMBL4604349

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human WM793 cells harboring BRAF V600E mutant assessed as reduction in cell viability after 24 hrs by EZ4U reagent based spectrophotometric method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type WM793
Confidence 1 — Organism
Curated By Autocuration

Target

WM793 (CHEMBL4630705)
Type CELL-LINE
Organism Homo sapiens

Publication

β,β-Dimethylacrylshikonin Induces Apoptosis in Melanoma Cell Lines by NOXA Upregulation.
Stallinger A, Kretschmer N, Kleinegger F, Brvar L, Liegl-Atzwanger B, Prokesch A, Durchschein C, Bauer R, Deutsch A, Rinner B.
J Nat Prod (2020) 83 : 305 -315
PubMed 31961147 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.92 5.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL267024 DIMETHYLACRYLSHIKONIN 1 5.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL267024 DIMETHYLACRYLSHIKONIN IC50 = 1200.0 nM 5.92