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Assay Detail

CHEMBL4604403

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against mouse B16F0 cells assessed as reduction in cell viability after 48 hrs by MTT assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type B16-F0
Confidence 1 — Organism
Curated By Autocuration

Target

B16-F0 (CHEMBL4296401)
Type CELL-LINE
Organism Mus musculus

Publication

β,β-Dimethylacrylshikonin Induces Apoptosis in Melanoma Cell Lines by NOXA Upregulation.
Stallinger A, Kretschmer N, Kleinegger F, Brvar L, Liegl-Atzwanger B, Prokesch A, Durchschein C, Bauer R, Deutsch A, Rinner B.
J Nat Prod (2020) 83 : 305 -315
PubMed 31961147 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.72 5.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL267024 DIMETHYLACRYLSHIKONIN 1 5.92
CHEMBL3327388 1 5.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL267024 DIMETHYLACRYLSHIKONIN IC50 = 1200.0 nM 5.92
CHEMBL3327388 IC50 = 3000.0 nM 5.52