Assay Detail
Functional
CHEMBL4606349
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antileishmanial activity against Leishmania major MON-4 intracellular amastigotes
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Leishmania major |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
O-Alkyl Hydroxamates Display Potent and Selective Antileishmanial Activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.01 | 6.02 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL935 | — | — | 1 | 6.02 |
| CHEMBL4640366 | — | — | 1 | 6.00 |
| CHEMBL239129 | MEGLUMINE ANTIMONATE | 3.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL935 | — | IC50 | = | 960.0 | nM | 6.02 |
| CHEMBL4640366 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL239129 | MEGLUMINE ANTIMONATE | IC50 | = | 101100.0 | nM | - |