Assay Detail
Functional
CHEMBL4610605
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Antiproliferative activity against human A549 cells assessed as reduction in cell growth measured after 72 hrs by Alamar blue assay
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | A549 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Rational design, synthesis and biological profiling of new KDM4C inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 5.79 | 7.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL578512 | — | — | 1 | 7.66 |
| CHEMBL1527391 | — | — | 1 | 5.96 |
| CHEMBL1517074 | — | — | 1 | 5.96 |
| CHEMBL4639254 | — | — | 1 | 5.89 |
| CHEMBL1438218 | — | — | 1 | 5.80 |
| CHEMBL4648732 | — | — | 1 | 5.72 |
| CHEMBL1316847 | — | — | 1 | 5.37 |
| CHEMBL4649004 | — | — | 1 | 5.24 |
| CHEMBL4646339 | — | — | 1 | 5.24 |
| CHEMBL4640783 | — | — | 1 | 5.06 |
| CHEMBL4640696 | — | — | 1 | - |
| CHEMBL1394266 | — | — | 1 | - |
| CHEMBL4636575 | — | — | 1 | - |
| CHEMBL4646564 | — | — | 1 | - |
| CHEMBL4640130 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL578512 | — | IC50 | = | 22.0 | nM | 7.66 |
| CHEMBL1527391 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL1517074 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL4639254 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL1438218 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL4648732 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL1316847 | — | IC50 | = | 4300.0 | nM | 5.37 |
| CHEMBL4649004 | — | IC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL4646339 | — | IC50 | = | 5700.0 | nM | 5.24 |
| CHEMBL4640783 | — | IC50 | = | 8800.0 | nM | 5.06 |
| CHEMBL4640696 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL1394266 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4636575 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4646564 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4640130 | — | IC50 | > | 30000.0 | nM | - |