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Assay Detail

CHEMBL4615239

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HCV with glycoprotein E1 F291V mutant infected in human Huh7.5 cells assessed as reduction in viral RNA levels incubated for 72 hrs by qRT-PCR analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

2-((4-Arylpiperazin-1-yl)methyl)benzonitrile Derivatives as Orally Available Inhibitors of Hepatitis C Virus with a Novel Mechanism of Action.
Jiang X, Tan J, Wang Y, Chen J, Li J, Jiang Z, Quan Y, Jin J, Li Y, Cen S, Li Y, Peng Z, Li Z.
J Med Chem (2020) 63 : 5972 -5989
PubMed 32378892 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.92 6.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4634954 1 6.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4634954 EC50 = 120.0 nM 6.92