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Assay Detail

CHEMBL4616990

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
In-vivo inhibition of beta-glucuronidase in BALB/CJ mouse at 10 ug administered as twice daily
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Beta-glucuronidase (CHEMBL4523185)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Therapeutic significance of β-glucuronidase activity and its inhibitors: A review.
Awolade P, Cele N, Kerru N, Gummidi L, Oluwakemi E, Singh P.
Eur J Med Chem (2020) 187 : 111921 -111921
PubMed 31835168 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.79 6.79

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3903683 1 6.79

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3903683 IC50 = 164.0 nM 6.79