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Assay Detail

CHEMBL4618184

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human C4-2 cells transfected with HA-tagged survivin assessed as reduction in cell viability measured after 72 hrs by methylene blue staining based assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type LNCaP C4-2
Confidence 1 — Organism
Curated By Autocuration

Target

LNCaP C4-2 (CHEMBL4296460)
Type CELL-LINE
Organism Homo sapiens

Publication

Synthesis and Identification of a Novel Lead Targeting Survivin Dimerization for Proteasome-Dependent Degradation.
Peery R, Kyei-Baffour K, Dong Z, Liu J, de Andrade Horn P, Dai M, Liu JY, Zhang JT.
J Med Chem (2020) 63 : 7243 -7251
PubMed 32421328 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.16 5.16

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4635753 1 5.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4635753 IC50 = 7000.0 nM 5.16