Assay Detail
Functional
CHEMBL4619676
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Inhibition of colony formation in human BE(2)-C cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BE(2)-C |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Characterization of Conformationally Constrained Benzanilide Scaffolds for Potent and Selective HDAC8 Targeting.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.60 | 5.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4637798 | — | — | 1 | 5.68 |
| CHEMBL2170177 | — | — | 1 | 5.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4637798 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL2170177 | — | IC50 | = | 3100.0 | nM | 5.51 |