Assay Detail
Binding
CHEMBL4621251
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Inhibition of Clostridium histolyticum collagenase using FALGPA as substrate by spectrophotometric method
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Hathewaya histolytica |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
<i>N</i>-Aryl-3-mercaptosuccinimides as Antivirulence Agents Targeting <i>Pseudomonas aeruginosa</i> Elastase and <i>Clostridium</i> Collagenases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.50 | 8.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL306726 | — | — | 1 | 8.30 |
| CHEMBL313776 | — | — | 1 | 6.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL306726 | — | Ki | = | 5.0 | nM | 8.30 |
| CHEMBL313776 | — | Ki | = | 200.0 | nM | 6.70 |