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Assay Detail

CHEMBL4627595

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against human HeLa cells assessed as inhibition of cell viability incubated for 24 hrs by resazurin dye based fluorescence analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

HeLa (CHEMBL399)
Type CELL-LINE
Organism Homo sapiens

Publication

Synthesis and biological evaluation of bis-N<sup>2</sup>,N<sup>2</sup>'-(4-hydroxycoumarin-3-yl)ethylidene]-2,3-dihydroxysuccinodihydrazides.
Manyeruke MH, Tshiwawa T, Hoppe HC, Isaacs M, Seldon R, Warner DF, Krause RWM, Kaye PT.
Bioorg Med Chem Lett (2020) 30 : 126911 -126911
PubMed 31952962 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.89 7.89

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL50588 EMETINE 4.0 1 7.89

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL50588 EMETINE IC50 = 13.0 nM 7.89