Assay Detail
Functional
CHEMBL4649946
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Leishmania donovani Ubiquitin Activating Enzyme (LdE1)
9165
Total Activities
8948
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Leishmania donovani |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Ubiquitin-activating enzyme e1, putative (CHEMBL4662923) ↗| Type | SINGLE PROTEIN |
| Organism | Leishmania donovani (strain BPK282A1) |
Publication
University of Dundee, Small-Polar-MMV Screening Library
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Percent Effect | 8841 | - | - |
| IC50 | 324 | 4.17 | 4.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3444410 | — | — | 3 | 4.35 |
| CHEMBL3443461 | — | — | 2 | 4.31 |
| CHEMBL3468912 | — | — | 3 | 4.30 |
| CHEMBL3443502 | — | — | 2 | 4.12 |
| CHEMBL3444390 | — | — | 3 | 4.07 |
| CHEMBL3443504 | — | — | 2 | 4.06 |
| CHEMBL3443503 | — | — | 2 | 4.04 |
| CHEMBL3493915 | — | — | 1 | - |
| CHEMBL3493934 | — | — | 1 | - |
| CHEMBL3493975 | — | — | 1 | - |
| CHEMBL3494069 | — | — | 1 | - |
| CHEMBL3495821 | — | — | 1 | - |
| CHEMBL3495860 | — | — | 1 | - |
| CHEMBL3493945 | — | — | 1 | - |
| CHEMBL3493952 | — | — | 1 | - |
| CHEMBL3495814 | — | — | 1 | - |
| CHEMBL3495885 | — | — | 1 | - |
| CHEMBL3494087 | — | — | 1 | - |
| CHEMBL3493899 | — | — | 1 | - |
| CHEMBL3495851 | — | — | 1 | - |
| CHEMBL3494068 | — | — | 1 | - |
| CHEMBL3493914 | — | — | 1 | - |
| CHEMBL3495858 | — | — | 1 | - |
| CHEMBL3493890 | — | — | 1 | - |
| CHEMBL3493874 | — | — | 1 | - |
| CHEMBL3495654 | — | — | 1 | - |
| CHEMBL3495608 | — | — | 1 | - |
| CHEMBL3495505 | — | — | 1 | - |
| CHEMBL3495701 | — | — | 1 | - |
| CHEMBL3495661 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3444410 | — | IC50 | = | 44966.76 | nM | 4.35 |
| CHEMBL3444410 | — | IC50 | = | 45341.23 | nM | 4.34 |
| CHEMBL3443461 | — | IC50 | = | 48535.79 | nM | 4.31 |
| CHEMBL3468912 | — | IC50 | = | 50324.1 | nM | 4.30 |
| CHEMBL3443461 | — | IC50 | = | 54773.9 | nM | 4.26 |
| CHEMBL3468912 | — | IC50 | = | 60439.46 | nM | 4.22 |
| CHEMBL3443502 | — | IC50 | = | 74997.63 | nM | 4.12 |
| CHEMBL3443502 | — | IC50 | = | 81460.67 | nM | 4.09 |
| CHEMBL3444390 | — | IC50 | = | 85802.22 | nM | 4.07 |
| CHEMBL3443504 | — | IC50 | = | 86354.51 | nM | 4.06 |
| CHEMBL3443504 | — | IC50 | = | 89732.93 | nM | 4.05 |
| CHEMBL3444390 | — | IC50 | = | 90964.34 | nM | 4.04 |
| CHEMBL3443503 | — | IC50 | = | 92200.55 | nM | 4.04 |
| CHEMBL3469953 | — | Percent Effect | = | 5.263 | % | - |
| CHEMBL3471855 | — | Percent Effect | = | 10.81 | % | - |
| CHEMBL3469629 | — | Percent Effect | = | 18.42 | % | - |
| CHEMBL3469676 | — | Percent Effect | = | 18.42 | % | - |
| CHEMBL3469692 | — | Percent Effect | = | -5.263 | % | - |
| CHEMBL3469891 | — | Percent Effect | = | 18.42 | % | - |
| CHEMBL3469814 | — | Percent Effect | = | 15.79 | % | - |
| CHEMBL3469845 | — | Percent Effect | = | 5.263 | % | - |
| CHEMBL3471750 | — | Percent Effect | = | 5.405 | % | - |
| CHEMBL3471753 | — | Percent Effect | = | 10.81 | % | - |
| CHEMBL3444400 | — | Percent Effect | = | 21.05 | % | - |
| CHEMBL3471702 | — | Percent Effect | = | 2.703 | % | - |
| CHEMBL3471728 | — | Percent Effect | = | 13.51 | % | - |
| CHEMBL3502468 | — | Percent Effect | = | -2.703 | % | - |
| CHEMBL3502465 | — | Percent Effect | = | 16.22 | % | - |
| CHEMBL3498473 | — | Percent Effect | = | 8.108 | % | - |
| CHEMBL3471747 | — | Percent Effect | = | 13.51 | % | - |
| CHEMBL3504226 | — | Percent Effect | = | 5.405 | % | - |
| CHEMBL3471760 | — | Percent Effect | = | 5.405 | % | - |
| CHEMBL3502369 | — | Percent Effect | = | - | % | - |
| CHEMBL3504179 | — | Percent Effect | = | 8.108 | % | - |
| CHEMBL3471716 | — | Percent Effect | = | 8.108 | % | - |
| CHEMBL3471765 | — | Percent Effect | = | 2.703 | % | - |
| CHEMBL3502484 | — | Percent Effect | = | - | % | - |
| CHEMBL3502481 | — | Percent Effect | = | 8.108 | % | - |
| CHEMBL3504195 | — | Percent Effect | = | 10.81 | % | - |
| CHEMBL3471712 | — | Percent Effect | = | 2.703 | % | - |
| CHEMBL3504229 | — | Percent Effect | = | - | % | - |
| CHEMBL3469821 | — | Percent Effect | = | 21.05 | % | - |
| CHEMBL3502475 | — | Percent Effect | = | 13.51 | % | - |
| CHEMBL3504186 | — | Percent Effect | = | 8.108 | % | - |
| CHEMBL3502471 | — | Percent Effect | = | 2.703 | % | - |
| CHEMBL3504227 | — | Percent Effect | = | -2.703 | % | - |
| CHEMBL3471722 | — | Percent Effect | = | 10.81 | % | - |
| CHEMBL3469943 | — | Percent Effect | = | 2.632 | % | - |
| CHEMBL3469699 | — | Percent Effect | = | 7.895 | % | - |
| CHEMBL3469807 | — | Percent Effect | = | 23.68 | % | - |