Assay Detail
Functional
CHEMBL4667670
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Antiproliferative activity against human OCILY3 cells by cell proliferation assay
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | OCI-Ly3 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Quinoline and thiazolopyridine allosteric inhibitors of MALT1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 28 | 5.94 | 6.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4748253 | — | — | 1 | 6.92 |
| CHEMBL4791759 | — | — | 1 | 6.57 |
| CHEMBL4784899 | — | — | 1 | 6.44 |
| CHEMBL4789469 | — | — | 1 | 6.39 |
| CHEMBL4779581 | — | — | 1 | 6.25 |
| CHEMBL4749826 | — | — | 1 | 6.23 |
| CHEMBL4790415 | — | — | 1 | 6.21 |
| CHEMBL4749854 | — | — | 1 | 6.14 |
| CHEMBL4751498 | — | — | 1 | 6.14 |
| CHEMBL4741853 | — | — | 1 | 6.14 |
| CHEMBL4740768 | — | — | 1 | 6.05 |
| CHEMBL4784740 | — | — | 1 | 6.00 |
| CHEMBL4794268 | — | — | 1 | 5.87 |
| CHEMBL4788571 | — | — | 1 | 5.84 |
| CHEMBL4763765 | — | — | 1 | 5.82 |
| CHEMBL4762086 | — | — | 1 | 5.80 |
| CHEMBL4740000 | — | — | 1 | 5.62 |
| CHEMBL4742156 | — | — | 1 | 5.62 |
| CHEMBL4755479 | — | — | 1 | 5.35 |
| CHEMBL4760252 | — | — | 1 | 5.15 |
| CHEMBL4782908 | — | — | 1 | 5.14 |
| CHEMBL4759864 | — | — | 1 | 4.89 |
| CHEMBL4780316 | — | — | 1 | - |
| CHEMBL4751202 | — | — | 1 | - |
| CHEMBL4784606 | — | — | 1 | - |
| CHEMBL4799622 | — | — | 1 | - |
| CHEMBL4777911 | — | — | 1 | - |
| CHEMBL4783451 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4748253 | — | EC50 | = | 120.0 | nM | 6.92 |
| CHEMBL4791759 | — | EC50 | = | 270.0 | nM | 6.57 |
| CHEMBL4784899 | — | EC50 | = | 360.0 | nM | 6.44 |
| CHEMBL4789469 | — | EC50 | = | 410.0 | nM | 6.39 |
| CHEMBL4779581 | — | EC50 | = | 560.0 | nM | 6.25 |
| CHEMBL4749826 | — | EC50 | = | 590.0 | nM | 6.23 |
| CHEMBL4790415 | — | EC50 | = | 620.0 | nM | 6.21 |
| CHEMBL4749854 | — | EC50 | = | 730.0 | nM | 6.14 |
| CHEMBL4751498 | — | EC50 | = | 730.0 | nM | 6.14 |
| CHEMBL4741853 | — | EC50 | = | 720.0 | nM | 6.14 |
| CHEMBL4740768 | — | EC50 | = | 900.0 | nM | 6.05 |
| CHEMBL4784740 | — | EC50 | = | 990.0 | nM | 6.00 |
| CHEMBL4794268 | — | EC50 | = | 1350.0 | nM | 5.87 |
| CHEMBL4788571 | — | EC50 | = | 1460.0 | nM | 5.84 |
| CHEMBL4763765 | — | EC50 | = | 1530.0 | nM | 5.82 |
| CHEMBL4762086 | — | EC50 | = | 1580.0 | nM | 5.80 |
| CHEMBL4740000 | — | EC50 | = | 2390.0 | nM | 5.62 |
| CHEMBL4742156 | — | EC50 | = | 2420.0 | nM | 5.62 |
| CHEMBL4755479 | — | EC50 | = | 4430.0 | nM | 5.35 |
| CHEMBL4760252 | — | EC50 | = | 7020.0 | nM | 5.15 |
| CHEMBL4782908 | — | EC50 | = | 7170.0 | nM | 5.14 |
| CHEMBL4759864 | — | EC50 | = | 12900.0 | nM | 4.89 |
| CHEMBL4780316 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL4751202 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL4784606 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL4799622 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL4777911 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL4783451 | — | EC50 | > | 20000.0 | nM | - |