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Assay Detail

CHEMBL4668397

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiproliferative activity against human TE-671 cells incubated for 36 hrs
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type TE-671
Confidence 1 — Organism
Curated By Autocuration

Target

TE-671 (CHEMBL615012)
Type CELL-LINE
Organism Homo sapiens

Publication

Colchicine Alkaloids and Synthetic Analogues: Current Progress and Perspectives.
Gracheva IA,Shchegravina ES,Schmalz HG,Beletskaya IP,Fedorov AY
J Med Chem (2020) 63 : 10618 -10651
PubMed 32432867 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 8.86 10.62

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL18981 THIOCOLCHICINE 1 10.62
CHEMBL153629 1 10.08
CHEMBL153052 1 5.88
CHEMBL357350 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL18981 THIOCOLCHICINE IC50 = 0.024 nM 10.62
CHEMBL153629 IC50 = 0.084 nM 10.08
CHEMBL153052 IC50 = 1320.0 nM 5.88
CHEMBL357350 IC50 = 0.001 nM -