Assay Detail
Binding
CHEMBL4668432
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Inhibition of calf brain tubulin by turbidimetry
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Colchicine Alkaloids and Synthetic Analogues: Current Progress and Perspectives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 6.03 | 6.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1985898 | — | — | 1 | 6.52 |
| CHEMBL4761265 | — | — | 1 | 6.48 |
| CHEMBL1171848 | — | — | 1 | 6.37 |
| CHEMBL4776771 | — | — | 1 | 6.33 |
| CHEMBL4764947 | — | — | 1 | 6.17 |
| CHEMBL4781477 | — | — | 1 | 5.64 |
| CHEMBL4756529 | — | — | 1 | 4.68 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1985898 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL4761265 | — | IC50 | = | 330.0 | nM | 6.48 |
| CHEMBL1171848 | — | IC50 | = | 430.0 | nM | 6.37 |
| CHEMBL4776771 | — | IC50 | = | 470.0 | nM | 6.33 |
| CHEMBL4764947 | — | IC50 | = | 670.0 | nM | 6.17 |
| CHEMBL4781477 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL4756529 | — | IC50 | = | 21000.0 | nM | 4.68 |