Assay Detail
Functional
CHEMBL4670184
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Antiproliferative activities against human U-251 cells by SRB assay
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | U-251 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Bioactive Alkaloids from the Actinomycete Actinoalloteichus sp. ZZ1866.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 4.90 | 5.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4791630 | — | — | 1 | 5.70 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 5.41 |
| CHEMBL4763301 | — | — | 1 | 5.24 |
| CHEMBL4754075 | — | — | 1 | 4.92 |
| CHEMBL4757657 | — | — | 1 | 4.92 |
| CHEMBL1928402 | — | — | 1 | 4.92 |
| CHEMBL4789230 | — | — | 1 | 4.89 |
| CHEMBL4784386 | — | — | 1 | 4.82 |
| CHEMBL4761582 | — | — | 1 | 4.77 |
| CHEMBL4756703 | — | — | 1 | 4.72 |
| CHEMBL4740296 | — | — | 1 | 4.57 |
| CHEMBL4748065 | — | — | 1 | 4.44 |
| CHEMBL4758385 | — | — | 1 | 4.44 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4791630 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 3900.0 | nM | 5.41 |
| CHEMBL4763301 | — | IC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL4754075 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL4757657 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL1928402 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL4789230 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL4784386 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL4761582 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL4756703 | — | IC50 | = | 19000.0 | nM | 4.72 |
| CHEMBL4740296 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL4748065 | — | IC50 | = | 36000.0 | nM | 4.44 |
| CHEMBL4758385 | — | IC50 | = | 36000.0 | nM | 4.44 |