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Assay Detail

CHEMBL4670429

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Binding
Agonist activity at PPARgamma (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Peroxisome proliferator-activated receptor gamma (CHEMBL235)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Photohormones Enable Optical Control of the Peroxisome Proliferator-Activated Receptor γ (PPARγ).
Hinnah K,Willems S,Morstein J,Heering J,Hartrampf FWW,Broichhagen J,Leippe P,Merk D,Trauner D
J Med Chem (2020) 63 : 10908 -10920
PubMed 32886507 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 8.83 8.83

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL434063 1 8.83

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL434063 EC50 = 1.47 nM 8.83