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Assay Detail

CHEMBL4673451

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimalarial activity against chloroquine sensitive Plasmodium falciparum
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

An epigrammatic status of the azole-based antimalarial drugs
Sharma, Mousmee, Prasher, Parteek
RSC Med Chem (2020) 11 : 184 -211
PubMed 33479627 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 6.70 6.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL157101 KETOCONAZOLE 4.0 1 6.70
CHEMBL104 CLOTRIMAZOLE 4.0 1 6.70
CHEMBL91 MICONAZOLE 4.0 1 6.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL157101 KETOCONAZOLE IC50 = 200.0 nM 6.70
CHEMBL104 CLOTRIMAZOLE IC50 = 200.0 nM 6.70
CHEMBL91 MICONAZOLE IC50 = 200.0 nM 6.70