Assay Detail
Functional
CHEMBL4673472
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Antiplasmodial activity against chloroquine sensitive Plasmodium falciparum FCR-3 infected in human erythrocytes incubated for 72 hrs by giemsa staining based assay
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Plasmodium falciparum |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
An epigrammatic status of the azole-based antimalarial drugs
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 14 | 8.40 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL174325 | — | — | 1 | 8.40 |
| CHEMBL426036 | — | — | 1 | 8.40 |
| CHEMBL353322 | — | — | 1 | 8.40 |
| CHEMBL4779036 | — | — | 1 | 8.40 |
| CHEMBL4763964 | — | — | 1 | 8.40 |
| CHEMBL174445 | — | — | 1 | 8.40 |
| CHEMBL4759011 | — | — | 1 | 8.40 |
| CHEMBL3091932 | — | — | 1 | 8.40 |
| CHEMBL4749430 | — | — | 1 | 8.40 |
| CHEMBL4762535 | — | — | 1 | 8.40 |
| CHEMBL4765178 | — | — | 1 | 8.40 |
| CHEMBL4759095 | — | — | 1 | 8.40 |
| CHEMBL4745515 | — | — | 1 | 8.40 |
| CHEMBL4798664 | — | — | 1 | 8.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL174325 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL426036 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL353322 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4779036 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4763964 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL174445 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4759011 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3091932 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4749430 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4762535 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4765178 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4759095 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4745515 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4798664 | — | EC50 | = | 4.0 | nM | 8.40 |