Assay Detail
Binding
CHEMBL4675293
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Non-covalent reversible inhibition of human CSE
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of a Bioactive Inhibitor with a New Scaffold for Cystathionine γ-Lyase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Inhibition | 1 | - | - |
| IC50 | 1 | 5.21 | 5.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4761159 | — | — | 1 | 5.21 |
| CHEMBL275938 | AURINTRICARBOXYLIC ACID | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4761159 | — | IC50 | = | 6200.0 | nM | 5.21 |
| CHEMBL275938 | AURINTRICARBOXYLIC ACID | Inhibition | - | % | - |