Assay Detail
Binding
CHEMBL4679740
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of Vgamma9Vdelta2 T cells proliferation incubated for 3 days by gamma delta TCR/PE-CD3+ antibody staining based FACS analysis
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | Vgamma9Vdelta2 T cell |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Butyrophilin subfamily 3 member A1 (CHEMBL4105758) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Synthesis and Metabolism of BTN3A1 Ligands: Studies on Modifications of the Allylic Alcohol.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 12 | 7.38 | 8.34 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4746099 | — | — | 1 | 8.34 |
| CHEMBL4088948 | — | — | 1 | 8.27 |
| CHEMBL4744593 | — | — | 1 | 8.10 |
| CHEMBL4745129 | — | — | 1 | 7.92 |
| CHEMBL4739889 | — | — | 1 | 7.70 |
| CHEMBL4743999 | — | — | 1 | 7.33 |
| CHEMBL4776906 | — | — | 1 | 7.33 |
| CHEMBL4780556 | — | — | 1 | 7.31 |
| CHEMBL4742284 | — | — | 1 | 6.10 |
| CHEMBL4172453 | — | — | 1 | 5.40 |
| CHEMBL4780307 | — | — | 1 | - |
| CHEMBL4746944 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4746099 | — | EC50 | = | 4.6 | nM | 8.34 |
| CHEMBL4088948 | — | EC50 | = | 5.4 | nM | 8.27 |
| CHEMBL4744593 | — | EC50 | = | 8.0 | nM | 8.10 |
| CHEMBL4745129 | — | EC50 | = | 12.0 | nM | 7.92 |
| CHEMBL4739889 | — | EC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4743999 | — | EC50 | = | 47.0 | nM | 7.33 |
| CHEMBL4776906 | — | EC50 | = | 47.0 | nM | 7.33 |
| CHEMBL4780556 | — | EC50 | = | 49.0 | nM | 7.31 |
| CHEMBL4742284 | — | EC50 | = | 790.0 | nM | 6.10 |
| CHEMBL4172453 | — | EC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL4780307 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4746944 | — | EC50 | > | 100000.0 | nM | - |