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Assay Detail

CHEMBL4685400

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]-ketanserin from recombinant human 5HT2A receptor expressed in CHOK1 cell membranes measured after 1 hr by microbeta counting method
37
Total Activities
37
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type CHO-K1
Subcellular Membrane
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

5-hydroxytryptamine receptor 2A (CHEMBL224)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Multifunctional 6-fluoro-3-[3-(pyrrolidin-1-yl)propyl]-1,2-benzoxazoles targeting behavioral and psychological symptoms of dementia (BPSD).
Bucki A,Marcinkowska M,Śniecikowska J,Zagórska A,Jamrozik M,Pawłowski M,Głuch-Lutwin M,Siwek A,Jakubczyk M,Pytka K,Jastrzębska-Więsek M,Partyka A,Wesołowska A,Mierzejewski P,Kołaczkowski M
Eur J Med Chem (2020) 191 : 112149 -112149
PubMed 32105980 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 37 8.78 9.61

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4759492 1 9.61
CHEMBL4753094 1 9.61
CHEMBL4747225 1 9.61
CHEMBL4763085 1 9.48
CHEMBL4764006 1 9.46
CHEMBL4754193 1 9.40
CHEMBL4793608 1 9.38
CHEMBL4785434 1 9.35
CHEMBL4754138 1 9.35
CHEMBL4748379 1 9.23
CHEMBL4764468 1 9.13
CHEMBL4751063 1 9.10
CHEMBL4747978 1 9.10
CHEMBL4744007 1 9.03
CHEMBL4779739 1 8.99
CHEMBL4782149 1 8.96
CHEMBL4776225 1 8.96
CHEMBL4762226 1 8.96
CHEMBL4749824 1 8.89
CHEMBL4784414 1 8.87
CHEMBL4741142 1 8.81
CHEMBL6437 MIANSERIN 4.0 1 8.72
CHEMBL4780470 1 8.55
CHEMBL4795995 1 8.50
CHEMBL4778418 1 8.41
CHEMBL4784228 1 8.38
CHEMBL4750664 1 8.37
CHEMBL4775997 1 8.28
CHEMBL4760655 1 8.27
CHEMBL4764557 1 8.24

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4759492 Ki = 0.2455 nM 9.61
CHEMBL4747225 Ki = 0.2455 nM 9.61
CHEMBL4753094 Ki = 0.2455 nM 9.61
CHEMBL4763085 Ki = 0.3311 nM 9.48
CHEMBL4764006 Ki = 0.3467 nM 9.46
CHEMBL4754193 Ki = 0.3981 nM 9.40
CHEMBL4793608 Ki = 0.4169 nM 9.38
CHEMBL4754138 Ki = 0.4467 nM 9.35
CHEMBL4785434 Ki = 0.4467 nM 9.35
CHEMBL4748379 Ki = 0.5888 nM 9.23
CHEMBL4764468 Ki = 0.7413 nM 9.13
CHEMBL4751063 Ki = 0.7943 nM 9.10
CHEMBL4747978 Ki = 0.7943 nM 9.10
CHEMBL4744007 Ki = 0.9333 nM 9.03
CHEMBL4779739 Ki = 1.023 nM 8.99
CHEMBL4782149 Ki = 1.096 nM 8.96
CHEMBL4762226 Ki = 1.096 nM 8.96
CHEMBL4776225 Ki = 1.096 nM 8.96
CHEMBL4749824 Ki = 1.288 nM 8.89
CHEMBL4784414 Ki = 1.349 nM 8.87
CHEMBL4741142 Ki = 1.549 nM 8.81
CHEMBL6437 MIANSERIN Ki = 1.905 nM 8.72
CHEMBL4780470 Ki = 2.818 nM 8.55
CHEMBL4795995 Ki = 3.162 nM 8.50
CHEMBL4778418 Ki = 3.89 nM 8.41
CHEMBL4784228 Ki = 4.169 nM 8.38
CHEMBL4750664 Ki = 4.266 nM 8.37
CHEMBL4775997 Ki = 5.248 nM 8.28
CHEMBL4760655 Ki = 5.37 nM 8.27
CHEMBL4764557 Ki = 5.754 nM 8.24
CHEMBL4750587 Ki = 6.457 nM 8.19
CHEMBL4790020 Ki = 8.913 nM 8.05
CHEMBL4742856 Ki = 9.12 nM 8.04
CHEMBL4763106 Ki = 9.55 nM 8.02
CHEMBL4758402 Ki = 11.48 nM 7.94
CHEMBL4796647 Ki = 15.49 nM 7.81
CHEMBL4748107 Ki = 19.5 nM 7.71