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Assay Detail

CHEMBL4685403

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]-methylspiperone from recombinant human D2 receptor expressed in CHOK1 cell membranes measured after 60 mins by microbeta counting method
37
Total Activities
37
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type CHO-K1
Subcellular Membrane
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

D(2) dopamine receptor (CHEMBL217)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Multifunctional 6-fluoro-3-[3-(pyrrolidin-1-yl)propyl]-1,2-benzoxazoles targeting behavioral and psychological symptoms of dementia (BPSD).
Bucki A,Marcinkowska M,Śniecikowska J,Zagórska A,Jamrozik M,Pawłowski M,Głuch-Lutwin M,Siwek A,Jakubczyk M,Pytka K,Jastrzębska-Więsek M,Partyka A,Wesołowska A,Mierzejewski P,Kołaczkowski M
Eur J Med Chem (2020) 191 : 112149 -112149
PubMed 32105980 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 37 7.89 9.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4747225 1 9.70
CHEMBL4795995 1 9.35
CHEMBL4747978 1 9.20
CHEMBL4759492 1 9.03
CHEMBL4764006 1 8.91
CHEMBL4754193 1 8.85
CHEMBL4748379 1 8.76
CHEMBL54 HALOPERIDOL 4.0 1 8.73
CHEMBL4760655 1 8.59
CHEMBL4744007 1 8.51
CHEMBL4753094 1 8.25
CHEMBL4751063 1 8.08
CHEMBL4780470 1 8.05
CHEMBL4742856 1 8.04
CHEMBL4785434 1 7.91
CHEMBL4763085 1 7.85
CHEMBL4778418 1 7.82
CHEMBL4764468 1 7.79
CHEMBL4762226 1 7.75
CHEMBL4793608 1 7.70
CHEMBL4754138 1 7.69
CHEMBL4784414 1 7.62
CHEMBL4750664 1 7.50
CHEMBL4776225 1 7.49
CHEMBL4763106 1 7.46
CHEMBL4749824 1 7.42
CHEMBL4790020 1 7.41
CHEMBL4782149 1 7.36
CHEMBL4775997 1 7.25
CHEMBL4764557 1 7.25

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4747225 Ki = 0.1995 nM 9.70
CHEMBL4795995 Ki = 0.4467 nM 9.35
CHEMBL4747978 Ki = 0.631 nM 9.20
CHEMBL4759492 Ki = 0.9333 nM 9.03
CHEMBL4764006 Ki = 1.23 nM 8.91
CHEMBL4754193 Ki = 1.413 nM 8.85
CHEMBL4748379 Ki = 1.738 nM 8.76
CHEMBL54 HALOPERIDOL Ki = 1.862 nM 8.73
CHEMBL4760655 Ki = 2.57 nM 8.59
CHEMBL4744007 Ki = 3.09 nM 8.51
CHEMBL4753094 Ki = 5.623 nM 8.25
CHEMBL4751063 Ki = 8.318 nM 8.08
CHEMBL4780470 Ki = 8.913 nM 8.05
CHEMBL4742856 Ki = 9.12 nM 8.04
CHEMBL4785434 Ki = 12.3 nM 7.91
CHEMBL4763085 Ki = 14.13 nM 7.85
CHEMBL4778418 Ki = 15.14 nM 7.82
CHEMBL4764468 Ki = 16.22 nM 7.79
CHEMBL4762226 Ki = 17.78 nM 7.75
CHEMBL4793608 Ki = 19.95 nM 7.70
CHEMBL4754138 Ki = 20.42 nM 7.69
CHEMBL4784414 Ki = 23.99 nM 7.62
CHEMBL4750664 Ki = 31.62 nM 7.50
CHEMBL4776225 Ki = 32.36 nM 7.49
CHEMBL4763106 Ki = 34.67 nM 7.46
CHEMBL4749824 Ki = 38.02 nM 7.42
CHEMBL4790020 Ki = 38.9 nM 7.41
CHEMBL4782149 Ki = 43.65 nM 7.36
CHEMBL4775997 Ki = 56.23 nM 7.25
CHEMBL4784228 Ki = 56.23 nM 7.25
CHEMBL4764557 Ki = 56.23 nM 7.25
CHEMBL4758402 Ki = 95.5 nM 7.02
CHEMBL4741142 Ki = 100.0 nM 7.00
CHEMBL4748107 Ki = 102.33 nM 6.99
CHEMBL4779739 Ki = 104.71 nM 6.98
CHEMBL4750587 Ki = 169.82 nM 6.77
CHEMBL4796647 Ki = 323.59 nM 6.49