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Assay Detail

CHEMBL4688558

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]-LSD from 5HT7 receptor (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

5-hydroxytryptamine receptor 7 (CHEMBL3155)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

A study of the structure-affinity relationship in SYA16263; is a D receptor interaction essential for inhibition of apormorphine-induced climbing behavior in mice?
Onyameh EK,Bricker BA,Eyunni SVK,Voshavar C,Gonela UM,Ofori E,Jenkins A,Ablordeppey SY
Bioorg Med Chem (2021) 30 : 115943 -115943
PubMed 33338898 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.05 7.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1940418 1 7.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1940418 Ki = 90.0 nM 7.05