Assay Detail
Functional
CHEMBL4699725
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human BJAB cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BJAB |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Application of triazoles as bioisosteres and linkers in the development of microtubule targeting agents
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.31 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4744630 | — | — | 1 | 8.40 |
| CHEMBL4744576 | — | — | 1 | 8.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4744630 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4744576 | — | IC50 | = | 6.0 | nM | 8.22 |