Assay Detail
Binding
CHEMBL4700002
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Mixed type inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by Dixon plot analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Tissue | Liver |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Synthesis, evaluation and molecular modelling of piceatannol analogues as arginase inhibitors
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 4.09 | 4.09 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4754674 | — | — | 1 | 4.09 |
| CHEMBL69863 | PICEATANNOL | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4754674 | — | Ki | = | 82000.0 | nM | 4.09 |
| CHEMBL69863 | PICEATANNOL | Ki | = | 136000.0 | nM | - |