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Assay Detail

CHEMBL4701319

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Phototoxicity against human SK-MEL-28 cells assessed as reduction in cell viability preincubated for 16 hrs followed by irradiated with 100 J/cm2 400 to 700 nanometer visible light for 40 mins and measured after 48 hrs by alamar blue assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type SK-MEL-28
Confidence 1 — Organism
Curated By Autocuration

Target

SK-MEL-28 (CHEMBL614919)
Type CELL-LINE
Organism Homo sapiens

Publication

Enhanced Production and Anticancer Properties of Photoactivated Perylenequinones.
Al Subeh ZY,Raja HA,Monro S,Flores-Bocanegra L,El-Elimat T,Pearce CJ,McFarland SA,Oberlies NH
J Nat Prod (2020) 83 : 2490 -2500
PubMed 32786877 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 6 7.25 7.99

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4796095 1 7.99
CHEMBL4793204 1 7.83
CHEMBL4792950 1 7.27
CHEMBL4748633 1 6.87
CHEMBL4786703 1 6.76
CHEMBL4787050 1 6.75

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4796095 EC50 = 10.3 nM 7.99
CHEMBL4793204 EC50 = 14.7 nM 7.83
CHEMBL4792950 EC50 = 53.5 nM 7.27
CHEMBL4748633 EC50 = 135.0 nM 6.87
CHEMBL4786703 EC50 = 172.0 nM 6.76
CHEMBL4787050 EC50 = 176.0 nM 6.75