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Assay Detail

CHEMBL4701355

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Functional
Antimalarial activity against chloroquine-sensitive Plasmodium falciparum HB3 assessed as reduction in [3H]-hypoxanthine incorporation pretreated for 24 hrs followed by [3H]-hypoxanthine addition measured after 24 hrs by liquid scintillation counting method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Structural hybridization as a facile approach to new drug candidates.
Sampath Kumar HM,Herrmann L,Tsogoeva SB
Bioorg Med Chem Lett (2020) 30 : 127514 -127514
PubMed 32860980 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 10.05 10.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL24704 1 10.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL24704 IC50 = 0.09 nM 10.05