Assay Detail
Functional
CHEMBL4702986
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Inhibition of LPS-induced NO production in mouse BV-2 cells
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | BV-2 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Anti-Inflammatory ent-Kaurane Diterpenoids from Isodon serra.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 11 | 4.79 | 5.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL356703 | — | — | 1 | 5.44 |
| CHEMBL4751286 | — | — | 1 | 5.14 |
| CHEMBL4755804 | — | — | 1 | 4.81 |
| CHEMBL4745397 | — | — | 1 | 4.58 |
| CHEMBL4789694 | — | — | 1 | 4.40 |
| CHEMBL4790884 | — | — | 1 | 4.36 |
| CHEMBL4752078 | — | — | 1 | - |
| CHEMBL4756539 | — | — | 1 | - |
| CHEMBL4760880 | — | — | 1 | - |
| CHEMBL4798923 | — | — | 1 | - |
| CHEMBL4761737 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL356703 | — | IC50 | = | 3600.0 | nM | 5.44 |
| CHEMBL4751286 | — | IC50 | = | 7300.0 | nM | 5.14 |
| CHEMBL4755804 | — | IC50 | = | 15600.0 | nM | 4.81 |
| CHEMBL4745397 | — | IC50 | = | 26200.0 | nM | 4.58 |
| CHEMBL4789694 | — | IC50 | = | 40100.0 | nM | 4.40 |
| CHEMBL4790884 | — | IC50 | = | 44100.0 | nM | 4.36 |
| CHEMBL4752078 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4756539 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4760880 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4798923 | — | IC50 | > | 60000.0 | nM | - |
| CHEMBL4761737 | — | IC50 | > | 100000.0 | nM | - |