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Assay Detail

CHEMBL4704735

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Dengue virus 2'-O methyltransferase incubated for 15 mins followed by [methyl-3-H]-AdoMet addition and measured after 30 mins by microbeta counter method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Dengue virus
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Synthesis and biological evaluation of novel flexible nucleoside analogues that inhibit flavivirus replication in vitro.
Thames JE,Waters CD,Valle C,Bassetto M,Aouadi W,Martin B,Selisko B,Falat A,Coutard B,Brancale A,Canard B,Decroly E,Seley-Radtke KL
Bioorg Med Chem (2020) 28 : 115713 -115713
PubMed 33128910 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.39 7.39

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1214186 SINEFUNGIN 2.0 1 7.39

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1214186 SINEFUNGIN IC50 = 41.0 nM 7.39