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Assay Detail

CHEMBL4706780

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of N-terminal His6-tagged Plasmodium falciparum DHODH expressed in Escherichia coli BL21 using L-DHO as substrate and CoQ as co-substrate by DCIP dye based spectrophotometric assay
34
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Plasmodium falciparum
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Tetrahydro-2-naphthyl and 2-Indanyl Triazolopyrimidines Targeting Plasmodium falciparum Dihydroorotate Dehydrogenase Display Potent and Selective Antimalarial Activity.
Kokkonda S,Deng X,White KL,Coteron JM,Marco M,de Las Heras L,White J,El Mazouni F,Tomchick DR,Manjalanagara K,Rudra KR,Chen G,Morizzi J,Ryan E,Kaminsky W,Leroy D,Martínez-Martínez MS,Jimenez-Diaz MB,Bazaga SF,Angulo-Barturen I,Waterson D,Burrows JN,Matthews D,Charman SA,Phillips MA,Rathod PK
J Med Chem (2016) 59 : 5416 -5431
PubMed 27127993 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 34 7.01 8.43

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4761666 2 8.43
CHEMBL4747214 2 8.34
CHEMBL4753862 2 8.34
CHEMBL4751920 1 8.20
CHEMBL1956285 DSM-265 2.0 1 8.05
CHEMBL4790441 1 7.85
CHEMBL4750037 2 7.82
CHEMBL4751321 1 7.68
CHEMBL4744317 2 7.68
CHEMBL4740960 1 7.62
CHEMBL4784152 1 7.32
CHEMBL4740342 1 7.28
CHEMBL4794107 1 7.28
CHEMBL4760917 2 7.22
CHEMBL4791257 1 7.19
CHEMBL4760735 1 7.18
CHEMBL4797521 1 7.11
CHEMBL4784677 1 7.07
CHEMBL4764319 1 7.06
CHEMBL4777941 1 7.05
CHEMBL4756700 1 6.96
CHEMBL4797946 1 6.92
CHEMBL4754938 1 6.85
CHEMBL4741128 1 6.85
CHEMBL3689094 1 6.77
CHEMBL4764723 1 6.10
CHEMBL4746414 1 5.40
CHEMBL4748163 1 5.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4761666 IC50 = 3.7 nM 8.43
CHEMBL4747214 IC50 = 4.6 nM 8.34
CHEMBL4753862 IC50 = 4.6 nM 8.34
CHEMBL4751920 IC50 = 6.3 nM 8.20
CHEMBL1956285 DSM-265 IC50 = 8.9 nM 8.05
CHEMBL4790441 IC50 = 14.0 nM 7.85
CHEMBL4750037 IC50 = 15.0 nM 7.82
CHEMBL4751321 IC50 = 21.0 nM 7.68
CHEMBL4744317 IC50 = 21.0 nM 7.68
CHEMBL4740960 IC50 = 24.0 nM 7.62
CHEMBL4784152 IC50 = 48.0 nM 7.32
CHEMBL4740342 IC50 = 52.0 nM 7.28
CHEMBL4794107 IC50 = 52.0 nM 7.28
CHEMBL4760917 IC50 = 60.0 nM 7.22
CHEMBL4791257 IC50 = 65.0 nM 7.19
CHEMBL4760735 IC50 = 66.0 nM 7.18
CHEMBL4797521 IC50 = 77.0 nM 7.11
CHEMBL4784677 IC50 = 85.0 nM 7.07
CHEMBL4764319 IC50 = 87.0 nM 7.06
CHEMBL4777941 IC50 = 89.0 nM 7.05
CHEMBL4756700 IC50 = 110.0 nM 6.96
CHEMBL4797946 IC50 = 120.0 nM 6.92
CHEMBL4754938 IC50 = 140.0 nM 6.85
CHEMBL4741128 IC50 = 140.0 nM 6.85
CHEMBL3689094 IC50 = 170.0 nM 6.77
CHEMBL4753862 IC50 = 640.0 nM 6.19
CHEMBL4747214 IC50 = 790.0 nM 6.10
CHEMBL4764723 IC50 = 790.0 nM 6.10
CHEMBL4744317 IC50 = 1000.0 nM 6.00
CHEMBL4750037 IC50 = 1100.0 nM 5.96
CHEMBL4761666 IC50 = 1340.0 nM 5.87
CHEMBL4760917 IC50 = 2300.0 nM 5.64
CHEMBL4746414 IC50 = 4000.0 nM 5.40
CHEMBL4748163 IC50 = 8000.0 nM 5.10